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Royal Society of Chemistry, RSC Medicinal Chemistry, 11(12), p. 1958-1967, 2021

DOI: 10.1039/d1md00025j

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Modulating β-arrestin 2 recruitment at the δ- and μ-opioid receptors using peptidomimetic ligands

Journal article published in 2021 by Krishna K. Sharma ORCID, Robert J. Cassell ORCID, Yazan J. Meqbil ORCID, Hongyu Su, Arryn T. Blaine ORCID, Benjamin R. Cummins, Kendall L. Mores ORCID, David K. Johnson ORCID, Richard M. van Rijn ORCID, Ryan A. Altman ORCID
This paper was not found in any repository, but could be made available legally by the author.
This paper was not found in any repository, but could be made available legally by the author.

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Abstract

C-Terminal modification of Leu-enkephalin analogs reduces β-arrestin signaling at the μ- and δ-opioid receptors. Such modifications will enable evaluation of novel signaling profiles for chronic pain management.