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Royal Society of Chemistry, MedChemComm, 9(10), p. 1646-1655, 2019

DOI: 10.1039/c9md00234k

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Piperidine carbamate peptidomimetic inhibitors of the serine proteases HGFA, matriptase and hepsin

Journal article published in 2019 by Vishnu C. Damalanka ORCID, Scott A. Wildman ORCID, James W. Janetka ORCID
This paper was not found in any repository, but could be made available legally by the author.
This paper was not found in any repository, but could be made available legally by the author.

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Abstract

A series of piperidine-based peptidomimetic inhibitors have been synthesized and evaluated their activity against the three serine proteases HGFA, matriptase, and hepsin. All analogs showed nanomolar activity against matriptase and hepsin.