Royal Society of Chemistry, MedChemComm, 5(10), p. 693-698, 2019
DOI: 10.1039/c9md00050j
Full text: Unavailable
The first syntheses of the bioactive cyclic tetrapeptide natural products, endolides A and B, were accomplished using a solution-phase macrocyclisation reaction; the stereoselectivity of which was found to be reagent-controlled.