Published in
Royal Society of Chemistry, MedChemComm, 9(7), p. 1793-1796
DOI: 10.1039/c6md00342g
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Design and synthesis of selective, small molecule inhibitors of coactivator-associated arginine methyltransferase 1 (CARM1)
Journal article published in 2016 by
H. Ü. Kaniskan,
M. S. Eram,
J. Liu,
D. Smil 
,
M. L. Martini,
Y. Shen,
V. Santhakumar,
P. J. Brown,
C. H. Arrowsmith,
M. Vedadi,
J. Jin
,
M. L. Martini,
Y. Shen,
V. Santhakumar,
P. J. Brown,
C. H. Arrowsmith,
M. Vedadi,
J. Jin
This paper is available in a repository.
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Abstract
Structure–activity relationship studies, starting from a fragment hit, resulted in discovery of the compound 9, an inhibitor of CARM1 with high potency and selectivity.