Joseph M. Hayes - Dissemin

All papers authored by Joseph M. Hayes

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2024 Levente Homolya

, Rachel T. Mathomes, Luca Varga, Tibor Docsa, László Juhász

, Joseph M. Hayes

, László Somsák

Synthesis, In Silico and Kinetics Evaluation of N-(β-d-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and N-(β-d-glucopyranosyl)-4(5)-arylimidazole-2-carboxamides as Glycogen Phosphorylase Inhibitors

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2023 Thomas D. Emmerich, Joseph M. Hayes

In Silico-Motivated Discovery of Novel Potent Glycogen Synthase-3 Inhibitors: 1-(Alkyl/arylamino)-3H-naphtho[1,2,3-de]quinoline-2,7-dione Identified as a Scaffold for Kinase Inhibitor Development

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Sándor Kun

, Rachel T. Mathomes

, Tibor Docsa, László Somsák

, Joseph M. Hayes

Design and Synthesis of 3-(β-d-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential

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2022 Mariann Kiss, István Timári, Teréz Barna, Zuzana Mészáros, Kristýna Slámová, Pavla Bojarová

, Vladimír Křen

, Joseph M. Hayes

, László Somsák

2-Acetamido-2-deoxy-d-glucono-1,5-lactone Sulfonylhydrazones: Synthesis and Evaluation as Inhibitors of Human OGA and HexB Enzymes

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Serafeim Alexopoulos, Anastasia Gkouskou, George Stravodimos, Anastasia S. Tsagkarakou, Ioannis Tsialtas, Demetres Katounis, Anna-Maria G. Psarra, Demetres Leonidas, Goutam Brahmachari, Joseph M. Hayes

, Vasiliki Skamnaki

The Druggability of the ATP Binding Site of Glycogen Phosphorylase Kinase Probed by Coumarin Analogues

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This paper was not found in any repository, but could be made available legally by the author.

2021 Christopher Lawson, Thowaiba Babikr Ahmed Alta, Georgia Moschou, Vasiliki Skamnaki

, Theodora G. A. Solovou, Caroline Topham

, Joseph Hayes

, Timothy J. Snape

Novel diarylamides and diarylureas with N-substitution dependent activity against medulloblastoma

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Mariann Kiss, Erna Szabó, Boglárka Bocska, Luu Thanh Sinh

, Conceicao Piedade Fernandes, István Timári, Joseph M. Hayes

, László Somsák

, Teréz Barna

Nanomolar inhibition of human OGA by 2-acetamido-2-deoxy-d-glucono-1,5-lactone semicarbazone derivatives

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Matthew P. Davies, Rocio Benitez, Concepción Perez, Sven Jakupovic, Philip Welsby, Klaudia Rzepecka, Jane Alder, Colin Davidson, Ana Martinez

, Joseph M. Hayes

Structure-Based Design of Potent Selective Nanomolar Type-II Inhibitors of Glycogen Synthase Kinase-3β

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2020 Ben A. Chetter, Efthimios Kyriakis, Daniel Barr, Aikaterini G. Karra, Elisabeth Katsidou, Symeon M. Koulas, Vassiliki T. Skamnaki, Timothy J. Snape, Anna-Maria G. Psarra, Demetres D. Leonidas, Joseph M. Hayes

Synthetic flavonoid derivatives targeting the glycogen phosphorylase inhibitor site: QM/MM-PBSA motivated synthesis of substituted 5,7-dihydroxyflavones, crystallography, in vitro kinetics and ex-vivo cellular experiments reveal novel potent inhibitors

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Jacek K. Wychowaniec

, Ronak Patel, James Leach, Rachel Mathomes, Vikesh Chhabria, Yogita Patil-Sen, Araida Hidalgo-Bastida, Robert T. Forbes, Joseph M. Hayes

, Mohamed A. Elsawy

Aromatic Stacking Facilitated Self-Assembly of Ultrashort Ionic Complementary Peptide Sequence: β-Sheet Nanofibers with Remarkable Gelation and Interfacial Properties

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2019 Daniel Barr, Eszter Szennyes, Éva Bokor, Ziad H. Al-Oanzi, Colin Moffatt, Sándor Kun, Tibor Docsa, Ádám Sipos, Matthew P. Davies, Rachel T. Mathomes, Timothy J. Snape

, Loranne Agius, László Somsák

, Joseph M. Hayes

Identification of C-β-d-Glucopyranosyl Azole-Type Inhibitors of Glycogen Phosphorylase That Reduce Glycogenolysis in Hepatocytes: In Silico Design, Synthesis, in Vitro Kinetics, and ex Vivo Studies

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Mark V. Sullivan, Sarah R. Dennison, Georgios Archontis, Subrayal M. Reddy

, Joseph M. Hayes

Toward Rational Design of Selective Molecularly Imprinted Polymers (MIPs) for Proteins: Computational and Experimental Studies of Acrylamide Based Polymers for Myoglobin

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2018 Aikaterini G. Karra, Maria Konstantinou

, Maria Tzortziou, Ioannis Tsialtas, Foteini D. Kalousi, Constantine Garagounis, Joseph M. Hayes

, Anna-Maria G. Psarra

Potential Dissociative Glucocorticoid Receptor Activity for Protopanaxadiol and Protopanaxatriol

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Sándor Kun, Jaida Begum, Efthimios Kyriakis, Evgenia C. V. Stamati, Thomas A. Barkas, Eszter Szennyes, Éva Bokor, Katalin E. Szabó, George A. Stravodimos, Ádám Sipos, Tibor Docsa, Pál Gergely, Colin Moffatt, Myrto S. Patraskaki

, Maria C. Kokolaki and 5 other authors

A multidisciplinary study of 3-(β- d -glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: Computation, synthesis, crystallography and kinetics reveal new potent inhibitors

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Demetra S. M. Chatzileontiadou

, Aikaterini C. Tsika, Zoi Diamantopoulou, Jean Delbé, Josette Badet, José Courty, Vassiliki T. Skamnaki, Vanessa Parmenopoulou, Dimitri Komiotis, Joseph M. Hayes

, Georgios A. Spyroulias, Demetres D. Leonidas

Evidence for Novel Action at the Cell‐Binding Site of Human Angiogenin Revealed by Heteronuclear NMR Spectroscopy, in silico and in vivo Studies

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2017 Demetres Leonidas, Joseph Hayes

, Atsushi Kato, Vassiliki Skamnaki, Demetra Chatzileontiadou

, Anastassia Kantsadi, Efthimios Kyriakis, Ben Chetter, George Stravodimos

Phytogenic Polyphenols as Glycogen Phosphorylase Inhibitors: The Potential of Triterpenes and Flavonoids for Glycaemic Control in Type 2 Diabetes

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Joseph M. Hayes

Computer-Aided Discovery of Glycogen Phosphorylase Inhibitors Exploiting Natural Products

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This paper is available in a repository.

2016 Demetra Georgatza, Vyron A. Gorgogietas, Paraskevi Kylindri, Maria C.-H. Charalambous

, Kalliope K. Papadopoulou

, Joseph M. Hayes

, Anna-Maria G. Psarra

The triterpene echinocystic acid and its 3-O-glucoside derivative are revealed as potent and selective glucocorticoid receptor agonists

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2015 Jaida Begum, Vassiliki T. Skamnaki, Colin Moffatt, Nicolas Bischler, Josephine Sarrou, Alexios-Leandros Skaltsounis, Demetres D. Leonidas, Nikos G. Oikonomakos, Joseph M. Hayes

An evaluation of indirubin analogues as phosphorylase kinase inhibitors

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Joseph M. Hayes

, Eric Deydier, Gregori Ujaque, Agustí Lledós, Raluca Malacea-Kabbara

, Eric Manoury, Sandrine Vincendeau, Rinaldo Poli

Ketone Hydrogenation with Iridium Complexes with “non N–H” Ligands: The Key Role of the Strong Base

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All papers authored by Joseph M. Hayes