Katarzyna Grychowska

All papers authored by Katarzyna Grychowska

This paper was not found in any repository, but could be made available legally by the author.

2023 Katarzyna Grychowska

, Uriel López-Sánchez, Mathieu Vitalis, Geoffrey Canet, Grzegorz Satała

, Agnieszka Olejarz-Maciej

, Joanna Gołębiowska, Rafał Kurczab, Wojciech Pietruś, Monika Kubacka, Christophe Moreau

, Maria Walczak

, Klaudia Blicharz-Futera

, Ophélie Bento, Xavier Bantreil

and 11 other authors

Superiority of the Triple-Acting 5-HT₆R/5-HT₃R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT₆R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats

Upload

2022 Katarzyna Grychowska

, Agnieszka Olejarz-Maciej

, Klaudia Blicharz, Wojciech Pietruś, Tadeusz Karcz, Rafał Kurczab, Paulina Koczurkiewicz, Agata Doroz-Płonka, Gniewomir Latacz, Abdul Raheem Keeri, Kamil Piska, Grzegorz Satała, Joanna Pęgiel, Wojciech Trybała, Magdalena Jastrzębska-Więsek and 8 other authors

Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines

Upload

2021 Paweł Zajdel

, Katarzyna Grychowska

, Szczepan Mogilski, Rafał Kurczab

, Grzegorz Satała

, Ryszard Bugno

, Tomasz Kos, Joanna Gołębiowska, Natalia Malikowska-Racia

, Agnieszka Nikiforuk

, Séverine Chaumont-Dubel

, Xavier Bantreil

, Maciej Pawłowski, Jean Martinez

, Gilles Subra

and 4 other authors

Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT₃ and 5-HT₆ Receptor Antagonist with Antipsychotic and Procognitive Properties

Upload

2020 Vittorio Canale, Katarzyna Grychowska

, Rafał Kurczab, Mateusz Ryng, Abdul Raheem Keeri, Grzegorz Satała, Agnieszka Olejarz-Maciej

, Paulina Koczurkiewicz, Marcin Drop

, Klaudia Blicharz, Kamil Piska, Elżbieta Pękala, Paulina Janiszewska, Martyna Krawczyk, Maria Walczak

and 5 other authors

A dual-acting 5-HT6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties

Upload

This paper is made freely available by the publisher.

Coralie Berthoux, Al Mahdy Hamieh, Angelina Rogliardo, Emilie L. Doucet, Camille Coudert, Fabrice Ango, Katarzyna Grychowska

, Séverine Chaumont‐Dubel, Pawel Zajdel, Rafael Maldonado, Joël Bockaert, Philippe Marin, Carine Bécamel

Early 5‐ HT 6 receptor blockade prevents symptom onset in a model of adolescent cannabis abuse

Download from onlinelibrary.wiley.com

2019 Katarzyna Grychowska

, Severine Chaumont-Dubel, Rafał Kurczab

, Paulina Koczurkiewicz, Caroline Deville, Martyna Krawczyk, Wojciech Pietruś, Grzegorz Satała, Szymon Buda, Kamil Piska, Marcin Drop, Xavier Bantreil

, Frédéric Lamaty

, Elżbieta Pękala, Andrzej J. Bojarski

and 3 other authors

Dual 5-HT6 and D3 Receptor Antagonists in a Group of 1H-Pyrrolo[3,2-c]quinolines with Neuroprotective and Procognitive Activity

Upload

2018 Katarzyna Grychowska

, Rafał Kurczab, Paweł Śliwa, Grzegorz Satała, Krzysztof Dubiel, Mikołaj Matłoka, Rafał Moszczyński-Pętkowski, Jerzy Pieczykolan, Andrzej J. Bojarski, Paweł Zajdel

Pyrroloquinoline scaffold-based 5-HT6R ligands: Synthesis, quantum chemical and molecular dynamic studies, and influence of nitrogen atom position in the scaffold on affinity

Upload

2017 Marcin Drop, Xavier Bantreil

, Katarzyna Grychowska

, Gilbert Umuhire Mahoro, Evelina Colacino, Maciej Pawłowski, Jean Martinez, Gilles Subra

, Pawel Zajdel, Frédéric Lamaty

Continuous flow ring-closing metathesis, an environmentally-friendly route to 2,5-dihydro-1H-pyrrole-3-carboxylates

Upload

2016 Katarzyna Grychowska

, Bartłomiej Kubica, Marcin Drop, Evelina Colacino, Xavier Bantreil, Maciej Pawłowski, Jean Martinez, Gilles Subra, Paweł Zajdel, Frédéric Lamaty

Application of the ring-closing metathesis to the formation of 2-aryl-1H-pyrrole-3-carboxylates as building blocks for biologically active compounds

Upload

Katarzyna Grychowska

, Grzegorz Satała, Tomasz Kos, Anna Partyka, Evelina Colacino, Severine Chaumont-Dubel, Xavier Bantreil, Anna Wesołowska, Maciej Pawłowski, Jean Martinez, Philippe Marin, Gilles Subra, Andrzej J. Bojarski, Frédéric Lamaty, Piotr Popik and 1 other authors

Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer’s Disease

Upload

2015 Beata Powroźnik, Karolina Słoczyńska, Vittorio Canale, Katarzyna Grychowska

, Paweł Zajdel, Elżbieta Pękala

Preliminary mutagenicity and genotoxicity evaluation of selected arylsulfonamide derivatives of (aryloxy)alkylamines with potential psychotropic properties

Upload

This paper is available in a repository.

Katarzyna Grychowska

, Nicolas Masurier, Pascal Verdie, Grzegorz Satała, Andrzej J. Bojarski, Jean Martinez, Maciej Pawłowski, Gilles Subra, Paweł Zajdel

Solid-Supported Synthesis and 5-HT7/5-HT1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1H)-one

Download from www.researchgate.net

2013 Katarzyna Grychowska

, Krzysztof Marciniec, Vittorio Canale, Michał Szymiec, Grzegorz Glanowski, Grzegorz Satała, Andrzej Maślankiewicz, Maciej Pawłowski, Andrzej J. Bojarski, Paweł Zajdel

Quinolinesulfonamides of Aryloxy‐/Arylthio‐ethyl Piperidines: Influence of an Arylether Fragment on 5‐HT_1A/5‐HT₇ Receptor Selectivity

Upload

Paweł Zajdel, Krzysztof Marciniec, Andrzej Maślankiewicz, Katarzyna Grychowska

, Grzegorz Satała, Beata Duszyńska, Tomasz Lenda, Agata Siwek, Gabriel Nowak, Anna Partyka

, Dagmara Wróbel, Magdalena Jastrzębska-Więsek, Andrzej J. Bojarski, Anna Wesołowska, Maciej Pawłowski

Antidepressant and antipsychotic activity of new quinoline- and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT1A/5-HT2A/5-HT7 and dopamine D2/D3 receptors

Download from www.researchgate.net

2012 Paweł Zajdel, Rafał Kurczab, Katarzyna Grychowska

, Grzegorz Satała, Maciej Pawłowski, Andrzej J. Bojarski

The multiobjective based design, synthesis and evaluation of the arylsulfonamide/amide derivatives of aryloxyethyl- and arylthioethyl- piperidines and pyrrolidines as a novel class of potent 5-HT7 receptor antagonists

Upload

2011 Paweł Zajdel, Joanna Król, Katarzyna Grychowska

, Maciej Pawłowski, Gilles Subra, Gaël Nomezine, Jean Martinez, Grzegorz Satała, Andrzej J. Bojarski, Ziniu Zhou, Martin J. O 'donnell, Martin J. O’Donnell, William L. Scott

Solid-Phase Synthesis of Arylpiperazine Derivatives and Implementation of the Distributed Drug Discovery (D3) Project in the Search for CNS Agents

Download from doi.org

Missing publications? Search for publications with a matching author name.

Researcher

Statistics

Refine

All papers authored by Katarzyna Grychowska