Hugo F. Costa-Almeida

All papers authored by Hugo F. Costa-Almeida

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Sara C. Silva Reis, Ivo E. Sampaio Dias, Daniela Correia da Silva, Xavier Cruz Correia, Hugo F. Costa-Almeida

, Beatriz L. Pires Lima, Vera Marisa Costa, A. L. Et

Discovery of Glypromate Conjugates with Biomedical Applications in Alzheimeir's Disease

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This paper is made freely available by the publisher.

Sara C. Silva-Reis

, Ivo E. Sampaio-Dias

, Vera M. Costa, Xavier Cruz Correia, Hugo F. Costa-Almeida

, Xerardo García-Mera, José E. Rodríguez-Borges

Concise Overview of Glypromate Neuropeptide Research: From Chemistry to Pharmacological Applications in Neurosciences

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Sara C. Silva Reis, Ivo E. Sampaio Dias, Xavier Cruz Correia, Hugo F. Costa Almeida

, Vera Marisa Costa, Daniela Correia da Silva, David M. Pereira, Xerardo García-Mera, José Enrique Rodriguez Borges

Glypromate Conjugates for Application in Neurodegenerative Diseases

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2022 Hugo F. Costa Almeida

, Ivo E. Sampaio Dias, Sara C. Silva Reis, Xavier Cruz Correia, Vera M. Costa, Félix D. Carvalho, Xerardo García-Mera, José E. Rodríguez Borges

Synthesis, Pharmacological and Toxicological Evaluation of Potent Melanostatin Peptidomimetics Incorporating Chiral β-Amino Acids as Proline Surrogates

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Hugo F. Costa Almeida

, Ivo E. Sampaio Dias, Sara C. Silva Reis, Xavier Cruz Correia, Vera M. Costa, Xerardo García-Mera, José E. Rodríguez Borges

Uma Abordagem Bioisostérica na Descoberta de Potentes Análogos da Melanostatina Usando β-Aminoácidos

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Xavier Cruz Correia, Ivo E. Sampaio Dias, Sara C. Silva Reis, Hugo F. Costa Almeida

, Vera M. Costa, Xerardo García-Mera, José E. Rodríguez Borges

Melanostatin Aza-Peptides as Potent Allosteric Modulators of the Dopamine D2 Receptors

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Sara C. Silva Reis, Ivo E. Sampaio Dias, Hugo F. Costa Almeida

, Vera M. Costa, Xerardo García-Mera, José E. Rodríguez Borges

A Chemical Strategy to Improve Bioavailability of Glypromate Peptide-Conjugates

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Sara C. Silva Reis, Ivo E. Sampaio Dias, Vera M. Costa, Xavier Cruz Correia, Hugo F. Costa Almeida

, Xerardo García-Mera, José E. Rodríguez Borges

Design, Synthesis, and Biological Evaluation of Glypromate-Based Neuroprotective Conjugates with Pharmaceutical Active Ingredients

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Sara C. Silva Reis, Ivo E. Sampaio Dias, Xavier Cruz Correia, Hugo F. Costa Almeida

, Vera M. Costa, Xerardo García-Mera, José E. Rodríguez Borges

Peptide-Amine Conjugates Targeting Neurodegenerative Diseases

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Sara C. Silva Reis, Ivo E. Sampaio Dias, Vera M. Costa, Xavier Cruz Correia, Hugo F. Costa Almeida

, Xerardo García-Mera, José E. Rodríguez Borges

Application of Hybrid Glypromate® Conjugates in Neurodegenerative Diseases

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Hugo F. Costa Almeida

, Ivo E. Sampaio Dias, Sara C. Silva Reis, Beatriz L. Pires Lima, Xavier Cruz Correia, Xerardo García-Mera, José E. Rodríguez Borges

Synthesis and Pharmacological Evaluation of Melanostatin Peptidomimetics Using β-Amino Acids as Proline Surrogates with Application in Parkinson’s Disease

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Beatriz L. Pires Lima, Ivo E. Sampaio Dias, Sara C. Silva Reis, Xavier Cruz Correia, Hugo F. Costa Almeida

, Xerardo García-Mera, José E. Rodríguez Borges

Triophene-Based Melanostatin (MIF-1) Neuropeptide Analogues by O-to-S Bioisosteric Replacement in MIF-1 Furoyl Peptidomimetics

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2021 Ivo E. Sampaio-Dias

, Sara C. Silva-Reis, Beatriz L. Pires-Lima

, Xavier Cruz Correia, Hugo F. Costa-Almeida

A Convenient On-Site Oxidation Strategy for the N-Hydroxylation of Melanostatin Neuropeptide Using Cope Elimination

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Hugo F. Costa-Almeida

, Sara C. Silva-Reis, Beatriz L. Pires-Lima, Ivo E. Sampaio-Dias, Xavier Cruz Correia, Xerardo García-Mera, José E. Rodríguez-Borges

Synthesis and pharmacological evaluation of melanostatin analogues containing Chiral β-amino acids as proline surrogates

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Beatriz L. Pires-Lima, Sara C. Silva-Reis, Xavier Cruz Correia, Xavier Cruz Correia, Ivo E. Sampaio-Dias, Hugo F. Costa-Almeida

, Xerardo García-Mera, José E. Rodriguéz-Borges

Exploring the bioisosterism of proline residue in melanostatin neuropeptide using heteroaromatic scaffolds

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Xavier Cruz Correia, Xavier Cruz Correia, Sara C. Silva-Reis, Beatriz L. Pires-Lima, Ivo E. Sampaio-Dias, Hugo F. Costa-Almeida

, Xerardo García-Mera, José E. Rodríguez-Borges

Using aza-proline for the assembly of a melanostatin aza-peptide derivative

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Sara C. Silva Reis, Ivo E. Sampaio Dias, Beatriz L. Pires Lima, Xavier Cruz Correia, Hugo F. Costa Almeida

, Xerardo García-Mera, José E. Rodríguez Borges

The Design of New Trofinetide® Conjugates Using Constrained Prolines

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Beatriz L. Pires Lima, Sara C. Silva Reis, Xavier Cruz Correia, Hugo F. Costa Almeida

, Xerardo García-Mera, José E. Rodríguez Borges, Ivo E. Sampaio Dias

Probing Heteroaromatic Scaffolds in the Melanostatin Neuropeptide: A Bioisosteric Approach Using Niacin as a Pro Surrogate

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Beatriz L. Pires Lima, Ivo E. Sampaio Dias, Sara C. Silva Reis, Xavier Cruz Correia, Hugo F. Costa Almeida

, Xerardo García-Mera, José E. Rodríguez Borges

Exploring the Role of the N-terminal Secondary Amine in Melanostatin Neuropeptide: A Bioisosteric Approach using (S)-Tetrahydro-2-furoic Acid as a Proline Surrogate

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All papers authored by Hugo F. Costa-Almeida