Joaquin Campos
investigacion.ugr.es
0000-0002-9035-8123
124 papers found
Refreshing results…
Actual Targets in Cytodifferentiation Cancer Therapy
Inhibition of choline kinase as a specific cytotoxic strategy in oncogene-transformed cells
Conformational Dynamics of a Bispyridinium Cyclophane
Neighbouring-group participation as the key step in the reactivity of acyclic and cyclic salicyl-derived O,O-acetals with 5-fluorouracil. Antiproliferative activity, cell cycle dysregulation and apoptotic induction of new O,N-acetals against breast cancer cells
QSAR-Derived Choline Kinase Inhibitors: How Rational can Antiproliferative Drug Design Be?
Medium benzene-fused oxacycles with the 5-fluorouracil moiety: synthesis, antiproliferative activities and apoptosis induction in breast cancer cells
Bispyridinium Cyclophanes: Novel Templates for Human Choline Kinase Inhibitors
Choline kinase inhibitory effect and antiproliferative activity of new 1,1 ' 1 ''-(benzene-1,3,5-triylmethylene)tris{4- (disubstituted)amino pyridinium } tribromides
Synthesis and spectral study of a novel distamycin conjugate
Quantitative structure–activity relationships for a series of symmetrical bisquaternary anticancer compounds
1H and13C chemical shifts for bis(benzopyridinium) dibromides with semirigid aromatic linkers
Identification of Novel Cyclooxygenase-2 Selective Inhibitors Using Pharmacophore Models
cis- and trans-1-[3-(Hydroxymethyl)-1,4-dioxepan-5-yl]pyrimidines: a new nucleoside prototype with a seven-membered moiety
LUMO energy of model compounds of bispyridinium compounds as an index for the inhibition of choline kinase
From a Classic Approach in Cancer Chemotherapy Towards Differentiation Therapy: Acyclic and Cyclic Seven-Membered 5-Fluorouracil O,N-Acetals
Modulation of myogenic differentiation in a human rhabdomyosarcoma cell line by a new derivative of 5-fluorouracil (QF-3602)
QSAR of 1,1′-(1,2-ethylenebisbenzyl)bis(4-substitutedpyridinium) dibromides as choline kinase inhibitors: a different approach for antiproliferative drug design
Synthesis, molecular modeling, and pharmacological testing of bis-quinolinium cyclophanes: Potent, non-peptidic blockers of the apamin-sensitive Ca2+-activated K+ channel
GR-891: a novel 5-fluorouracil acyclonucleoside prodrug for differentiation therapy in rhabdomyosarcoma cells
Synthesis of novel 5-fluorouracil derivatives with 1,4-oxaheteroepane moieties
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