Rob Leurs
0000-0003-1354-2848
10 papers found
Refreshing results…
Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H1 Receptor
Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics
Label-Free Analysis with Multiple Parameters Separates G Protein-Coupled Receptor Signaling Pathways
Development of a conformational histamine H3 receptor biosensor for the synchronous screening of agonists and inverse agonists.
A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light
Route to Prolonged Residence Time at the Histamine H1 Receptor: Growing from Desloratadine to Rupatadine
Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity
A Photoswitchable Agonist for the Histamine H 3 Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor
Photoswitching the Efficacy of a Small-Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism
Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity
Missing publications? Search for publications with a matching author name.