Giovanni Grazioso

Papers authored by Giovanni Grazioso

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2011 Clelia Dallanoce

, Fabio Frigerio, Giovanni Grazioso

, Carlo Matera

, Giacomo Luca Visconti, Marco De Amici

, Luca Pucci, Francesco Pistillo, Sergio Fucile, Cecilia Gotti, Francesco Clementi, Carlo De Micheli

New spirocyclic Δ2-isoxazoline derivatives related to selective agonists of α7 neuronal nicotinic acetylcholine receptors

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Giovanni Grazioso

, Vittorio Limongelli, Davide Branduardi, Ettore Novellino, Carlo De Micheli, Andrea Cavalli, Michele Parrinello

Investigating the Mechanism of Substrate Uptake and Release in the Glutamate Transporter Homologue Glt(Ph) through Metadynamics Simulations

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Luca Pucci, Giovanni Grazioso

, Clelia Dallanoce, Luca Rizzi, Carlo De Micheli, Francesco Clementi, Sonia Bertrand, Daniel Bertrand, Renato Longhi, Marco De Amici, Cecilia Gotti

Engineering of α-conotoxin MII-derived peptides with increased selectivity for native α6β2* nicotinic acetylcholine receptors

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Roberta Ettari, Maria Zappalà, Nicola Micale, Giovanni Grazioso

, Salvatore Giofrè, Tanja Schirmeister, Silvana Grasso

Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors

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Clelia Dallanoce

, Pietro Magrone, Carlo Matera

, Fabio Frigerio, Giovanni Grazioso

, Marco De Amici

, Sergio Fucile, Vanessa Piccari, Karla Frydenvang, Luca Pucci, Cecilia Gotti, Francesco Clementi, Carlo De Micheli

Design, Synthesis, and Pharmacological Characterization of Novel Spirocyclic Quinuclidinyl-Δ2-Isoxazoline Derivatives as Potent and Selective Agonists of α7 Nicotinic Acetylcholine Receptors

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Andrea Pinto, Paola Conti

, Giovanni Grazioso

, Lucia Tamborini

, Ulf Madsen, Birgitte Nielsen, Carlo De Micheli

Synthesis of new isoxazoline-based acidic amino acids and investigation of their affinity and selectivity profile at ionotropic glutamate receptors

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Laura Legnani, Federica Compostella, Giovanni Grazioso

, Franca Marinone Albini, Lucio Toma

Molecular dynamics simulations of the Salmonella typhi Vi antigenic polysaccharide and effects of the introduction of a zwitterionic motif

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2010 Clelia Dallanoce

, Fabio Frigerio, Giuliana Martelli, Giovanni Grazioso

, Carlo Matera

, Diego Yuri Pomè, Luca Pucci, Francesco Clementi, Cecilia Gotti, Marco De Amici

Novel tricyclic Δ2-isoxazoline and 3-oxo-2-methyl-isoxazolidine derivatives: Synthesis and binding affinity at neuronal nicotinic acetylcholine receptor subtypes

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Gabriella Roda, Clelia Dallanoce

, Giovanni Grazioso

, Vincenzo Liberti, Marco De Amici

, Marco De Amici

Determination of Acid Dissociation Constants of Compounds Active at Neuronal Nicotinic Acetylcholine Receptors by Means of Electrophoretic and Potentiometric Techniques

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2009 Giovanni Grazioso

, Diego Yuri Pomè, Carlo Matera

, Fabio Frigerio, Luca Pucci, Cecilia Gotti, Clelia Dallanoce

, Marco De Amici

Design of novel α7-subtype-preferring nicotinic acetylcholine receptor agonists: Application of docking and MM-PBSA computational approaches, synthetic and pharmacological studies

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Jacopo Sgrignani

, Claudia Bonaccini, Giovanni Grazioso

, Matteo Chioccioli, Andrea Cavalli, Paola Gratteri

Insights into docking and scoring neuronal α4β2 nicotinic receptor agonists using molecular dynamics simulations and QM/MM calculations

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Maria Luisa Calabrò, Daniela Raneri, Paola Ficarra, Tiziana Mennini, Simona Colleoni, Giovanni Grazioso

, Nicola Micale, Maria Zappalà, Silvana Grasso

Synthesis, Chiral Resolution and Pharmacological Evaluation of a 2,3-Benzodiazepine-Derived Noncompetitive AMPA Receptor Antagonist

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Clelia Dallanoce

, Pietro Magrone, Paola Bazza, Giovanni Grazioso

, Luca Rizzi, Loredana Riganti, Cecilia Gotti, Francesco Clementi, Karla Frydenvang, Marco De Amici

New Analogues of Epiboxidine Incorporating the 4,5-Dihydroisoxazole Nucleus: Synthesis, Binding Affinity at Neuronal Nicotinic Acetylcholine Receptors, and Molecular Modeling Investigations

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2008 Giovanni Grazioso

, Andrea Cavalli, Marco De Amici

, Maurizio Recanatini, Carlo De Micheli

Alpha7 nicotinic acetylcholine receptor agonists: Prediction of their binding affinity through a molecular mechanics Poisson-Boltzmann surface area approach

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Andrea Pinto, Paola Conti

, Marco De Amici

, Lucia Tamborini

, Giovanni Grazioso

, Simona Colleoni, Tiziana Mennini, Marco Gobbi, Carlo De Micheli

Synthesis of enantiomerically pure HIP-A and HIP-B and investigation of their activity as inhibitors of excitatory amino acid transporters

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2007 Paola Conti

, Andrea Pinto, Lucia Tamborini

, Giovanni Grazioso

, Giovambattista De Sarro, Hans Bräuner-Osborne

, Geza Szabo, László Gábor Hársing, Carlo De Micheli

Synthesis of Conformationally Constrained Glutamic Acid Homologues and Investigation of Their Pharmacological Profiles

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2006 Paola Conti

, Marco De Amici

, Andrea Pinto, Lucia Tamborini

, Giovanni Grazioso

, Bente Frølund, Birgitte Nielsen, Christian Thomsen, Bjarke Ebert, Carlo De Micheli

Synthesis of 3-Hydroxy- and 3-Carboxy-Δ2-isoxazoline Amino Acids and Evaluation of Their Interaction with GABA Receptors and Transporters

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Clelia Dallanoce

, Paola Bazza, Giovanni Grazioso

, Marco De Amici

, Cecilia Gotti, Loredana Riganti, Francesco Clementi, Carlo De Micheli

Synthesis of Epibatidine-Related Δ2-Isoxazoline Derivatives and Evaluation of Their Binding Affinity at Neuronal Nicotinic Acetylcholine Receptors

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2005 Maria Zappalà, Giovanna Postorino, Nicola Micale, Salvatore Caccamese, Nunziatina Parrinello, Giovanni Grazioso

, Gabriella Roda, Frank S. Menniti, Giovambattista De Sarro, Silvana Grasso

Synthesis, Chiral Resolution, and Enantiopharmacology of a Potent 2,3-Benzodiazepine Derivative as Noncompetitive AMPA Receptor Antagonist

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Paola Conti

, Marco De Amici

, Giovanni Grazioso

, Gabriella Roda, Andrea Pinto, Kasper Bø Hansen, Birgitte Nielsen, Ulf Madsen, Hans Bräuner-Osborne

, Jan Egebjerg, Valentina Vestri, Domenico E. Pellegrini-Giampietro, Pauline Sibille, Francine C. Acher, Carlo De Micheli

Synthesis, Binding Affinity at Glutamic Acid Receptors, Neuroprotective Effects, and Molecular Modeling Investigation of Novel Dihydroisoxazole Amino Acids †

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Papers authored by Giovanni Grazioso