Published in
American Chemical Society, Journal of Medicinal Chemistry, 23(57), p. 9945-9957, 2014
DOI: 10.1021/jm5011622
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Indolylarylsulfones Carrying a Heterocyclic Tail as Very Potent and Broad Spectrum HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors
Journal article published in 2014 by
Valeria Famiglini,
Giuseppe La Regina,
Antonio Coluccia 
,
Sveva Pelliccia ,
Andrea Brancale,
Giovanni Maga,
Emmanuele Crespan,
Roger Badia,
Eva Riveira-Muñoz,
José A. Esté,
Rosella Ferretti,
Roberto Cirilli,
Claudio Zamperini,
Maurizio Botta,
Dominique Schols
and other authors.
,
Sveva Pelliccia ,
Andrea Brancale,
Giovanni Maga,
Emmanuele Crespan,
Roger Badia,
Eva Riveira-Muñoz,
José A. Esté,
Rosella Ferretti,
Roberto Cirilli,
Claudio Zamperini,
Maurizio Botta,
Dominique Schols
and other authors.
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Abstract
We synthesized new indolylarylsulfone (IAS) derivatives carrying a heterocyclic tail at the indole-2-carboxamide nitrogen as potential anti-HIV/AIDS agents. Several new IASs yielded EC50 values