Published in

Wiley-VCH Verlag, ChemInform, 6(44), p. no-no, 2013

DOI: 10.1002/chin.201306166

Wiley, Angewandte Chemie International Edition, 37(51), p. 9220-9222, 2012

DOI: 10.1002/anie.201205079

Links

Tools

Export citation

Search in Google Scholar

Efficient and Versatile Synthesis of Indoles from Enamines and Imines by Cross-Dehydrogenative Coupling

Journal article published in 2012 by Zhuangzhi Shi ORCID, Frank Glorius ORCID
This paper is available in a repository.
This paper is available in a repository.

Full text: Download

Red circle
Preprint: archiving forbidden
Orange circle
Postprint: archiving restricted
Upload
Red circle
Published version: archiving forbidden
Policy details
Data provided by SHERPA/RoMEO

Abstract

Complement for Fischer: An efficient palladium-catalyzed indole synthesis proceeds by the intramolecular cross-dehydrogenative coupling of N-aryl imines under mild conditions using molecular oxygen as the sole oxidant. This practical method relies on anilines and ketones as starting materials (and thus the same retrosynthetic disconnection as the Fischer indole synthesis) and will likely become a popular route.