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Elsevier, Tetrahedron, 44(58), p. 8947-8955

DOI: 10.1016/s0040-4020(02)01159-6

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Synthesis and nucleophilic opening of a new C2 symmetric bis-aziridine. First synthesis of aziridines using polymer-supported triphenylphosphine

Journal article published in 2002 by Isabelle McCort ORCID, Stéphanie Ballereau, Annie Duréault, Jean-Claude Depezay
This paper was not found in any repository, but could be made available legally by the author.
This paper was not found in any repository, but could be made available legally by the author.

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Abstract

The synthesis of (2S,2′S)-2,3-bis(aziridin-2-yl)quinoxaline 4 from d-mannitol is reported. Reductive aminocyclization of diazidodiols has been achieved by polymer-supported PPh3 in a suitable manner. The N-Boc and N-Tos aziridines 4b and 4c have been reacted with different nucleophiles either in protic or aprotic media.