Wiley-VCH Verlag, ChemInform, 16(43), p. no-no, 2012
Elsevier, Tetrahedron Letters, 52(52), p. 7157-7160
DOI: 10.1016/j.tetlet.2011.10.123
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A facile and operationally simple route to diastereomerically pure, natural-like 3-azabicyclo[3.3.1]non-6-enes via microwave-assisted, BF3·OEt2-promoted aza-Prins reaction has been developed. Complexity-generating transformations based on these products involving reactive functionalities introduced during the aza-Prins step have been developed.