Published in
Royal Society of Chemistry, Chemical Science, 12(12), p. 4519-4525, 2021
DOI: 10.1039/d0sc05442a
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Rapid Synthesis of Pomalidomide-Conjugates for the Development of Protein Degrader Libraries
Journal article published in 2021 by
Duncan Keith Brownsey 
,
Ben Christopher Rowley ,
Evgueni Gorobets ,
Benjamin Sidney Gelfand ,
Darren Jason Derksen
,
Ben Christopher Rowley ,
Evgueni Gorobets ,
Benjamin Sidney Gelfand ,
Darren Jason Derksen
This paper is made freely available by the publisher.
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Abstract
Current methods for the preparation of heterobifunctional pomalidomide-conjugates rely on methods that are often low yielding and produce intractable byproducts. Herein we describe our strategy for the succinct preparation of pomalidomide-linkers.