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Royal Society of Chemistry, Chemical Science, 14(10), p. 4069-4076, 2019

DOI: 10.1039/c8sc03669a

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Ligand discrimination between active and inactive activation loop conformations of Aurora-A kinase is unmodified by phosphorylation

Journal article published in 2019 by James A. H. Gilburt ORCID, Paul Girvan ORCID, Julian Blagg ORCID, Liming Ying ORCID, Charlotte A. Dodson ORCID
This paper is made freely available by the publisher.
This paper is made freely available by the publisher.

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Abstract

Activation loop phosphorylation changes the position of equilibrium between DFG-in-like and DFG-out-like conformations but not the conformational preference of inhibitors.