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Beilstein-Institut, Beilstein Journal of Organic Chemistry, (5), 2009

DOI: 10.3762/bjoc.5.36

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Dipyridodiazepinone derivatives; synthesis and anti HIV-1 activity

Journal article published in 2009 by Nisachon Khunnawutmanotham, Nitirat Chimnoi, Arunee Thitithanyanont, Patchreenart Saparpakorn, Kiattawee Choowongkomon, Pornpan Pungpo, Supa Hannongbua ORCID, Supanna Techasakul
This paper is made freely available by the publisher.
This paper is made freely available by the publisher.

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Abstract

Ten dipyridodiazepinone derivatives were synthesized and evaluated for their anti HIV-1 reverse transcriptase activity against wild-type and mutant type enzymes, K103N and Y181C. Two of them were found to be promising inhibitors for HIV-1 RT.