Masakazu Atobe - Dissemin

All papers authored by Masakazu Atobe

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2018 Masakazu Atobe

, Kenji Naganuma, Masashi Kawanishi, Takahiko Hayashi, Hiroko Suzuki, Masahiro Nishida, Hirokazu Arai

Discovery of a novel 2-(1 H -pyrazolo[3,4- b ]pyridin-1-yl)thiazole derivative as an EP 1 receptor antagonist and in vivo studies in a bone fracture model

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2017 John F. Darby

, Masakazu Atobe

, James D. Firth

, Paul Bond

, Gideon J. Davies

, Peter O'Brien

, Roderick E. Hubbard

Increase of enzyme activity through specific covalent modification with fragments

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2015 Monique Lüthy, Mary C. Wheldon, Chehasnah Haji-Cheteh, Masakazu Atobe

, Paul S. Bond

, Peter O'Brien, Roderick E. Hubbard, Ian J. S. Fairlamb

Lead-oriented synthesis: Investigation of organolithium-mediated routes to 3-D scaffolds and 3-D shape analysis of a virtual lead-like library

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2014 Masakazu Atobe

, Kenji Naganuma, Masashi Kawanishi, Akifumi Morimoto, Ken-Ichi Kasahara, Shigeki Ohashi, Hiroko Suzuki, Takahiko Hayashi, Shiro Miyoshi

Discovery of 2-(1H-indazol-1-yl)-thiazole derivatives as selective EP1 receptor antagonists for treatment of overactive bladder by core structure replacement

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Shinya Sogame, Yoshihito Suenaga, Masakazu Atobe

, Masashi Kawanishi, Eiichi Tanaka, Shiro Miyoshi

Discovery of a benzimidazole series of ADAMTS-5 (aggrecanase-2) inhibitors by scaffold hopping

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2013 Masakazu Atobe

, Kenji Naganuma, Masashi Kawanishi, Akifumi Morimoto, Ken-Ichi Kasahara, Shigeki Ohashi, Hiroko Suzuki, Takahiko Hayashi, Shiro Miyoshi

Hit-to-lead optimization of 2-(1H-pyrazol-1-yl)-thiazole derivatives as a novel class of EP1 receptor antagonists

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Masakazu Atobe

, Naomi Maekawara, Masashi Kawanishi, Hiroko Suzuki, Eiichi Tanaka, Shiro Miyoshi

Design, synthesis and SAR investigation of thienosultam derivatives as ADAMTS-5 (aggrecanase-2) inhibitors

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Masakazu Atobe

, Naomi Maekawara, Noriko Ishiguro, Shinya Sogame, Yoshihito Suenaga, Masashi Kawanishi, Hiroko Suzuki, Norimasa Jinno, Eiichi Tanaka, Shiro Miyoshi

A series of thiazole derivatives bearing thiazolidin-4-one as non-competitive ADAMTS-5 (aggrecanase-2) inhibitors

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2009 Naoki Yamazaki, Sakae Aoyagi, Masakazu Atobe

, Chihiro Kibayashi

New Entry to the Asymmetric Synthesis of (–)-Lasubine I and (+)-Subcosine I

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2005 Masakazu Atobe

, Naoki Yamazaki, Chihiro Kibayashi

Asymmetric synthesis of (+)-abresoline

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2004 Masakazu Atobe

, Naoki Yamazaki, Chihiro Kibayashi

Enantioselective Synthesis of Primary 1-(Aryl)alkylamines by Nucleophilic 1,2-Addition of Organolithium Reagents to Hydroxyoxime Ethers and Application to Asymmetric Synthesis of G-Protein-Coupled Receptor Ligands

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2002 Naoki Yamazaki, Masakazu Atobe

, Chihiro Kibayashi

Enantioselective synthesis of NK-1 receptor antagonists (+)-CP-99,994 and (+)-CP-122,721

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2001 Naoki Yamazaki, Masakazu Atobe

, Chihiro Kibayashi

Nucleophilic addition of methyllithium to chiral oxime ethers: asymmetric preparation of 1-(aryl)ethylamines and application to a synthesis of calcimimetics (+)-NPS R-568 and its thio analogue

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All papers authored by Masakazu Atobe